Activity record

PGDB_A080009

Assay: % DegradationTarget: CDK2QC: standardized
Activity overview

Dmax = 58.7 %

TargetCDK2
Cell lineHEK293T
Concentration10 uM
Assay / Readoutluminescence / Dmax
Assay IDPGDB_AS000752
PatentWO2026064643A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C030650
Compound IDPGDB_C030650
Compound1
Source record IDPGDB_C030650
InChIKeyUUYPPKYXJFUVSW-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000752
Assay family% Degradation
Assay systemcell_based
ReadoutDmax
Technologyluminescence
Concentration10 uM
TargetCDK2
E3Not specified
Cell lineHEK293T
OrganismHomo sapiens

Source evidence

Patent IDWO2026064643A1
Compound location

1

1 enlarged structure1 location on patent page 107
Activity table
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