Activity record

PGDB_A080480

Assay: viabilityTarget: ARQC: standardized
Activity overview

IC50 = 0.33 nM

TargetAR
Cell lineVCaP
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000271
PatentWO2026061104A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C030132
Compound IDPGDB_C030132
CompoundAR-P-458
Source record IDPGDB_C030132
InChIKeyULNPCBVBGMLFHZ-UVNRZBLTSA-N

Assay context

Assay IDPGDB_AS000271
Assay familyviability
Assay systemcell_based
ReadoutIC50
Detection target% Cell viability
TargetAR
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2026061104A1
Compound location

AR-P-458

AR-P-458 enlarged structureAR-P-458 location on patent page 258
Activity table
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