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Compound
PGDB_C030132
6 activity records1 related patents
2D structure
N#Cc1ccc(N2C(C(F)(F)F)CC23CCN(c2ccc(C(=O)N4CCC(CN5CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4=O)cc2)CC3)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 79 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000072 | PGDB_C030132 | PGDB_AS001072 | View |
| % Degradation | - | = | 3 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078528 | PGDB_C030132 | PGDB_AS002389 | View |
| % Degradation | - | = | 39 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A079849 | PGDB_C030132 | PGDB_AS001281 | View |
| IC50 | - | = | 1.43 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080479 | PGDB_C030132 | PGDB_AS000195 | View |
| IC50 | - | = | 0.33 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A080480 | PGDB_C030132 | PGDB_AS000271 | View |