Assay
PGDB_AS000060
System: biochemicalTarget: CRBN | DDB1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.011 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A014887 | PGDB_C006039 | PGDB_AS000060 | View | |
| IC50 | - | = | 0.043 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A020923 | PGDB_C006037 | PGDB_AS000060 | View | |
| IC50 | - | = | 0.052 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A032897 | PGDB_C006035 | PGDB_AS000060 | View | |
| IC50 | - | = | 0.009 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A036684 | PGDB_C006034 | PGDB_AS000060 | View | |
| IC50 | - | = | 0.018 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A037015 | PGDB_C006038 | PGDB_AS000060 | View | |
| IC50 | - | = | 0.024 | uM | - | — | CRBN | CRBN | - | AU2024222626A1 | PGDB_A076142 | PGDB_C006036 | PGDB_AS000060 | View |