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SIMM · NJU
Assay
PGDB_AS000086
System: cell_based
Cell line: KP4
Assay context summary
Assay context
250 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
E3
Not specified
Cell line
KP4
Technology
Western_blot
Detection target
protein_degradation
Activity compounds and values
Activity records
250 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A007378
PGDB_C023945
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A007647
PGDB_C023865
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A008169
PGDB_C024065
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A008455
PGDB_C023991
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A008658
PGDB_C024041
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009148
PGDB_C024026
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009439
PGDB_C024034
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009767
PGDB_C023938
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009789
PGDB_C023992
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009826
PGDB_C024066
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009865
PGDB_C023930
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A009881
PGDB_C024073
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A010207
PGDB_C024057
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A010385
PGDB_C023869
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A010389
PGDB_C024010
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A011122
PGDB_C024056
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A011473
PGDB_C023857
PGDB_AS000086
View
% Degradation
-
<
10
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A011521
PGDB_C024003
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A011537
PGDB_C023915
PGDB_AS000086
View
% Degradation
-
>=
70
%
0.1 uM
6 h
ELAVL1
-
KP4
CN120303269A
PGDB_A011877
PGDB_C023896
PGDB_AS000086
View