Assay
PGDB_AS000093
System: cell_basedCell line: MKN45
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ymin | - | = | 9.38 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A007527 | PGDB_C012569 | PGDB_AS000093 | View | |
| Ymin | - | = | 22.54 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A007542 | PGDB_C012555 | PGDB_AS000093 | View | |
| Ymin | - | = | 8.08 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A008762 | PGDB_C012521 | PGDB_AS000093 | View | |
| Ymin | - | = | 11.2 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A009529 | PGDB_C012564 | PGDB_AS000093 | View | |
| Ymin | - | = | 28.19 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A010125 | PGDB_C012509 | PGDB_AS000093 | View | |
| Ymin | - | = | 18.64 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A011314 | PGDB_C012543 | PGDB_AS000093 | View | |
| Ymin | - | = | 11.94 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A012377 | PGDB_C012517 | PGDB_AS000093 | View | |
| Ymin | - | = | 9.67 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A013165 | PGDB_C012550 | PGDB_AS000093 | View | |
| Ymin | - | = | 10.54 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A013481 | PGDB_C012512 | PGDB_AS000093 | View | |
| Ymin | - | = | 17.2 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A014286 | PGDB_C012505 | PGDB_AS000093 | View | |
| Ymin | - | = | 22.05 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A015363 | PGDB_C012485 | PGDB_AS000093 | View | |
| Ymin | - | = | 24.76 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A015724 | PGDB_C012520 | PGDB_AS000093 | View | |
| Ymin | - | = | 16.24 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A018074 | PGDB_C012510 | PGDB_AS000093 | View | |
| Ymin | - | = | 7.81 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A018234 | PGDB_C012486 | PGDB_AS000093 | View | |
| Ymin | - | = | 13.21 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A018464 | PGDB_C012568 | PGDB_AS000093 | View | |
| Ymin | - | = | 11.71 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A020347 | PGDB_C012534 | PGDB_AS000093 | View | |
| Ymin | - | = | 8.65 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A021058 | PGDB_C012508 | PGDB_AS000093 | View | |
| Ymin | - | = | 27.73 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A021844 | PGDB_C012539 | PGDB_AS000093 | View | |
| Ymin | - | = | 7.1 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A022893 | PGDB_C012522 | PGDB_AS000093 | View | |
| Ymin | - | = | 6.08 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A023299 | PGDB_C012496 | PGDB_AS000093 | View |