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Compound
PGDB_C012509
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(O[C@H]4CCN(Cc5cnn(-c6cccc(C(F)(F)F)c6)c5)C4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ymin | - | = | 28.19 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A010125 | PGDB_C012509 | PGDB_AS000093 | View |
| EC50 | - | = | 0.117 | uM | - | — | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A017165 | PGDB_C012509 | PGDB_AS002574 | View |
| Ymin | - | = | 31.08 | % | Concentration series: 1 uM, 10 uM | 4 h | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A018787 | PGDB_C012509 | PGDB_AS000656 | View |
| EC50 | - | = | 0.013 | uM | - | — | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A066164 | PGDB_C012509 | PGDB_AS000951 | View |