Assay
PGDB_AS000263
System: cell_basedCell line: THLE-2
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 150 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A038764 | PGDB_C001020 | PGDB_AS000263 | View | |
| IC50 | - | > | 150 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A049141 | PGDB_C001019 | PGDB_AS000263 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A051133 | PGDB_C001018 | PGDB_AS000263 | View | |
| IC50 | - | > | 150 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A066966 | PGDB_C001022 | PGDB_AS000263 | View | |
| IC50 | - | > | 150 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A072678 | PGDB_C001023 | PGDB_AS000263 | View | |
| IC50 | - | > | 150 | nM | - | — | GSPT1 | - | THLE-2 | CN121219280A | PGDB_A075873 | PGDB_C001021 | PGDB_AS000263 | View |