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SIMM · NJU
Assay
PGDB_AS000333
System: cell_based
Target: UBE2M
Cell line: KBM7
Assay context summary
Assay context
66 activity records
Assay family
viability
System
cell_based
Readout
EC50
Target
UBE2M
E3
Not specified
Cell line
KBM7
Organism
Homo sapiens
Technology
luminescence
Detection target
% Cell viability
Activity compounds and values
Activity records
66 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A007794
PGDB_C019085
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A012507
PGDB_C019086
PGDB_AS000333
View
EC50
-
=
1-10
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A014725
PGDB_C019107
PGDB_AS000333
View
EC50
-
=
1-10
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A015458
PGDB_C019094
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A015774
PGDB_C019135
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A016584
PGDB_C019145
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A016778
PGDB_C019144
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A019023
PGDB_C019117
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A019549
PGDB_C019138
PGDB_AS000333
View
EC50
-
=
0.25-0.5
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A020501
PGDB_C019136
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A021755
PGDB_C019114
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A022392
PGDB_C019099
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A022879
PGDB_C019091
PGDB_AS000333
View
EC50
-
=
1-10
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A023852
PGDB_C019096
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A023932
PGDB_C019130
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A025526
PGDB_C019129
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A027187
PGDB_C019142
PGDB_AS000333
View
EC50
-
>
10
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A028117
PGDB_C019093
PGDB_AS000333
View
EC50
-
=
0.5-1
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A028474
PGDB_C019110
PGDB_AS000333
View
EC50
-
<=
0.25
uM
-
—
-
-
KBM7
AU2021359129A1
PGDB_A028648
PGDB_C019126
PGDB_AS000333
View