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SIMM · NJU
Assay
PGDB_AS000413
System: cell_based
Cell line: K562
Assay context summary
Assay context
54 activity records
Assay family
viability
System
cell_based
Readout
GI50
E3
Not specified
Cell line
K562
Organism
Homo sapiens
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
54 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A007844
PGDB_C011978
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A008850
PGDB_C011990
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A009394
PGDB_C012019
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A010822
PGDB_C012024
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A010850
PGDB_C011972
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A011658
PGDB_C011974
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A012831
PGDB_C012020
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A013731
PGDB_C011983
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A014417
PGDB_C011988
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A014946
PGDB_C011998
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A015157
PGDB_C012003
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A015183
PGDB_C012006
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A015744
PGDB_C012027
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A016076
PGDB_C012028
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A017484
PGDB_C011989
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A017590
PGDB_C012022
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A018246
PGDB_C012021
PGDB_AS000413
View
GI50
-
<
1000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A020863
PGDB_C012029
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A021419
PGDB_C011986
PGDB_AS000413
View
GI50
-
>
3000
nM
-
—
CCNK
-
K562
WO2025245472A1
PGDB_A026358
PGDB_C012007
PGDB_AS000413
View