Assay
PGDB_AS000603
System: cell_basedTarget: KCNH2Cell line: HEK293
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | % Inhibition | - | = | 37.69 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A007639 | PGDB_C005388 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 60.74 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A009294 | PGDB_C005427 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 11.7 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A009743 | PGDB_C005413 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 52.8 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A010543 | PGDB_C005432 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 60.94 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A011423 | PGDB_C005423 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 16.23 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A011684 | PGDB_C005429 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 20.59 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A014065 | PGDB_C005390 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 48.92 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A015678 | PGDB_C005434 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 45.18 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A018419 | PGDB_C005410 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 24.56 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A018665 | PGDB_C005438 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 69.97 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A021350 | PGDB_C005447 | PGDB_AS000603 | View |
 | % Inhibition | - | = | -0.31 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A021584 | PGDB_C005402 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 40.62 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A022635 | PGDB_C005385 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 13.03 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A022970 | PGDB_C005421 | PGDB_AS000603 | View |
 | % Inhibition | - | = | -1.37 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A026631 | PGDB_C005436 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 40.69 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A026657 | PGDB_C005405 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 26.98 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A029993 | PGDB_C005442 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 13.24 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A030562 | PGDB_C005415 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 55.77 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A030585 | PGDB_C005387 | PGDB_AS000603 | View |
 | % Inhibition | - | = | 21.21 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A033168 | PGDB_C005407 | PGDB_AS000603 | View |