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SIMM · NJU
Assay
PGDB_AS000761
System: cell_based
Target: NEK7
Cell line: CAL-51
Assay context summary
Assay context
148 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
NEK7
E3
CRBN
Cell line
CAL-51
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
148 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A007238
PGDB_C020340
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A008045
PGDB_C020401
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A008352
PGDB_C020335
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A009445
PGDB_C020326
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A009587
PGDB_C026287
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A010005
PGDB_C020366
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A010990
PGDB_C020434
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A011178
PGDB_C020355
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A011277
PGDB_C020424
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A012523
PGDB_C020405
PGDB_AS000761
View
DC50
-
>
1000
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A012707
PGDB_C020292
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A012722
PGDB_C020351
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A012905
PGDB_C020284
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014087
PGDB_C020331
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014311
PGDB_C020312
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014379
PGDB_C020348
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014458
PGDB_C020389
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A015403
PGDB_C020287
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A015789
PGDB_C020374
PGDB_AS000761
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A017224
PGDB_C020423
PGDB_AS000761
View