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SIMM · NJU
Assay
PGDB_AS000913
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
136 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
136 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
45.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A007262
PGDB_C011348
PGDB_AS000913
View
Dmax
-
=
56.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A007268
PGDB_C011366
PGDB_AS000913
View
Dmax
-
=
52.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A007710
PGDB_C011363
PGDB_AS000913
View
Dmax
-
=
52
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A007921
PGDB_C011290
PGDB_AS000913
View
Dmax
-
=
47.7
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A007945
PGDB_C011292
PGDB_AS000913
View
Dmax
-
=
52.3
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A008883
PGDB_C011399
PGDB_AS000913
View
Dmax
-
=
41.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A009336
PGDB_C011396
PGDB_AS000913
View
Dmax
-
=
56.4
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A009401
PGDB_C011316
PGDB_AS000913
View
Dmax
-
=
40.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A009415
PGDB_C011322
PGDB_AS000913
View
Dmax
-
=
46.3
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A011192
PGDB_C011319
PGDB_AS000913
View
Dmax
-
=
55.8
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A011782
PGDB_C011390
PGDB_AS000913
View
Dmax
-
=
51.4
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A012314
PGDB_C011297
PGDB_AS000913
View
Dmax
-
=
31.5
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A012877
PGDB_C011341
PGDB_AS000913
View
Dmax
-
=
52
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A013070
PGDB_C011317
PGDB_AS000913
View
Dmax
-
=
49.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A014426
PGDB_C011352
PGDB_AS000913
View
Dmax
-
=
50.6
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A015635
PGDB_C011386
PGDB_AS000913
View
Dmax
-
=
43.2
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A015891
PGDB_C011382
PGDB_AS000913
View
Dmax
-
=
57.1
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A017173
PGDB_C011369
PGDB_AS000913
View
Dmax
-
=
60.3
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A017331
PGDB_C011387
PGDB_AS000913
View
Dmax
-
=
36.3
%
-
-
CDK2
-
HEK293
WO2025181261A1
PGDB_A018280
PGDB_C011343
PGDB_AS000913
View