Assay
PGDB_AS000997
System: cell_basedCell line: MKN45
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ymin | - | = | 10.5 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A007602 | PGDB_C011149 | PGDB_AS000997 | View | |
| Ymin | - | = | 83.5 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A007744 | PGDB_C011210 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.7 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A008532 | PGDB_C011145 | PGDB_AS000997 | View | |
| Ymin | - | = | 10.6 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A009124 | PGDB_C011105 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.5 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A009875 | PGDB_C011188 | PGDB_AS000997 | View | |
| Ymin | - | = | 11.2 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A009979 | PGDB_C011123 | PGDB_AS000997 | View | |
| Ymin | - | = | 15.5 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A010458 | PGDB_C011175 | PGDB_AS000997 | View | |
| Ymin | - | = | 13.4 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A010510 | PGDB_C011140 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.7 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A011072 | PGDB_C011206 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.9 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A011188 | PGDB_C011237 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.9 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A012027 | PGDB_C011139 | PGDB_AS000997 | View | |
| Ymin | - | = | 89.6 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A012382 | PGDB_C011202 | PGDB_AS000997 | View | |
| Ymin | - | = | 12.1 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A012588 | PGDB_C011106 | PGDB_AS000997 | View | |
| Ymin | - | = | 16.3 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A012988 | PGDB_C011239 | PGDB_AS000997 | View | |
| Ymin | - | = | 80.2 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A013872 | PGDB_C011232 | PGDB_AS000997 | View | |
| Ymin | - | = | 7.8 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A015159 | PGDB_C011143 | PGDB_AS000997 | View | |
| Ymin | - | = | 10.4 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A015708 | PGDB_C011201 | PGDB_AS000997 | View | |
| Ymin | - | = | 7.8 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A015841 | PGDB_C011206 | PGDB_AS000997 | View | |
| Ymin | - | = | 9.9 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A016542 | PGDB_C011116 | PGDB_AS000997 | View | |
| Ymin | - | = | 8.8 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2025137053A1 | PGDB_A018084 | PGDB_C011124 | PGDB_AS000997 | View |