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SIMM · NJU
Assay
PGDB_AS001094
System: biochemical
Target: CRBN | DDB1
Assay context summary
Assay context
205 activity records
Assay family
ternary_complex
System
biochemical
Readout
Emax
Target
CRBN | DDB1
E3
CRBN | DDB1
Activity compounds and values
Activity records
205 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A007573
PGDB_C012421
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A007649
PGDB_C012407
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A007730
PGDB_C012471
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A007769
PGDB_C012450
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A007980
PGDB_C012439
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A008220
PGDB_C012342
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A008497
PGDB_C012301
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A008890
PGDB_C012462
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A008961
PGDB_C012406
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A009123
PGDB_C012330
PGDB_AS001094
View
Emax
-
<
50
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A009203
PGDB_C012339
PGDB_AS001094
View
Emax
-
<
50
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A009356
PGDB_C012283
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A009407
PGDB_C012319
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A009810
PGDB_C012391
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A010327
PGDB_C012377
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A010398
PGDB_C012433
PGDB_AS001094
View
Emax
-
>
120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A011013
PGDB_C012320
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A011021
PGDB_C012280
PGDB_AS001094
View
Emax
-
=
50-120
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A011131
PGDB_C012375
PGDB_AS001094
View
Emax
-
<
50
%
-
2 h
ALK
CRBN
-
WO2026015344A1
PGDB_A011293
PGDB_C012363
PGDB_AS001094
View