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Cc1nc2ccc(-c3noc(CN4CCCC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)n3)cc2o1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | < | 50 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A009203 | PGDB_C012339 | PGDB_AS001094 | View | |
| EC50 | - | = | 10-100 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A023213 | PGDB_C012339 | PGDB_AS002152 | View | |
| EC50 | - | = | 100-1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A025117 | PGDB_C012339 | PGDB_AS000738 | View | |
| Emax | - | > | 120 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A062883 | PGDB_C012339 | PGDB_AS001769 | View |