Assay

PGDB_AS001106

System: cell_basedTarget: IKZF1Cell line: 293GT
Assay context summary

Assay context

28 activity records
Assay family% Degradation
Systemcell_based
ReadoutEC50
TargetIKZF1
E3Not specified
Cell line293GT
Detection targetprotein_degradation
Activity compounds and values

Activity records

28 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008952
EC50-=0.051uM-—IKZF1-293GTKR20210031923APGDB_A014323PGDB_C008952PGDB_AS001106View
2D structure for PGDB_C008940
EC50->50uM-—IKZF1-293GTKR20210031923APGDB_A014915PGDB_C008940PGDB_AS001106View
2D structure for PGDB_C008958
EC50-=0.57uM-—IKZF1-293GTKR20210031923APGDB_A015973PGDB_C008958PGDB_AS001106View
2D structure for PGDB_C008948
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A017362PGDB_C008948PGDB_AS001106View
2D structure for PGDB_C008955
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A018307PGDB_C008955PGDB_AS001106View
2D structure for PGDB_C008963
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A018851PGDB_C008963PGDB_AS001106View
2D structure for PGDB_C008960
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A019090PGDB_C008960PGDB_AS001106View
2D structure for PGDB_C008953
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A019126PGDB_C008953PGDB_AS001106View
2D structure for PGDB_C008941
EC50->50uM-—IKZF1-293GTKR20210031923APGDB_A021266PGDB_C008941PGDB_AS001106View
2D structure for PGDB_C008945
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A024051PGDB_C008945PGDB_AS001106View
2D structure for PGDB_C008954
EC50-=0.63uM-—IKZF1-293GTKR20210031923APGDB_A024999PGDB_C008954PGDB_AS001106View
2D structure for PGDB_C008944
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A025531PGDB_C008944PGDB_AS001106View
2D structure for PGDB_C008937
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A027450PGDB_C008937PGDB_AS001106View
2D structure for PGDB_C008946
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A029081PGDB_C008946PGDB_AS001106View
2D structure for PGDB_C008959
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A035676PGDB_C008959PGDB_AS001106View
2D structure for PGDB_C008949
EC50-=0.12uM-—IKZF1-293GTKR20210031923APGDB_A038291PGDB_C008949PGDB_AS001106View
2D structure for PGDB_C008712
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A038939PGDB_C008712PGDB_AS001106View
2D structure for PGDB_C008961
EC50-=2.37uM-—IKZF1-293GTKR20210031923APGDB_A039819PGDB_C008961PGDB_AS001106View
2D structure for PGDB_C008942
EC50->50uM-—IKZF1-293GTKR20210031923APGDB_A047973PGDB_C008942PGDB_AS001106View
2D structure for PGDB_C008956
EC50->30uM-—IKZF1-293GTKR20210031923APGDB_A048668PGDB_C008956PGDB_AS001106View
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