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SIMM · NJU
Assay
PGDB_AS001171
System: biochemical
Target: BTRC | FBXW11 | SKP1
Assay context summary
Assay context
128 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
BTRC | FBXW11 | SKP1
E3
BTRC | FBXW11 | SKP1
Activity compounds and values
Activity records
128 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007347
PGDB_C021012
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A008167
PGDB_C021088
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A008437
PGDB_C021074
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A008997
PGDB_C021016
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009070
PGDB_C021017
PGDB_AS001171
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009676
PGDB_C021081
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010363
PGDB_C021062
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010401
PGDB_C021064
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010788
PGDB_C021068
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010984
PGDB_C021067
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A011417
PGDB_C021084
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012405
PGDB_C021024
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013306
PGDB_C021110
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013979
PGDB_C021116
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A014289
PGDB_C021048
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A014839
PGDB_C021060
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A014848
PGDB_C021055
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015344
PGDB_C021063
PGDB_AS001171
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015531
PGDB_C021061
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A017756
PGDB_C021030
PGDB_AS001171
View