Assay
PGDB_AS001228
System: cell_basedCell line: VCaP
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | VCaP | CN116239566A | PGDB_A011012 | PGDB_C025826 | PGDB_AS001228 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | VCaP | CN116239566A | PGDB_A036240 | PGDB_C025824 | PGDB_AS001228 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | VCaP | CN116239566A | PGDB_A039319 | PGDB_C019597 | PGDB_AS001228 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | VCaP | CN116239566A | PGDB_A055246 | PGDB_C025823 | PGDB_AS001228 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | VCaP | CN116239566A | PGDB_A072439 | PGDB_C019596 | PGDB_AS001228 | View |