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SIMM · NJU
Assay
PGDB_AS001244
System: cell_based
Target: IKZF2
Cell line: 293GT
Assay context summary
Assay context
181 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF2
E3
Not specified
Cell line
293GT
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
181 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.002
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A007134
PGDB_C008799
PGDB_AS001244
View
EC50
-
=
0.085
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A007708
PGDB_C008841
PGDB_AS001244
View
EC50
-
=
0.018
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009126
PGDB_C008771
PGDB_AS001244
View
EC50
-
=
0.077
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009132
PGDB_C008830
PGDB_AS001244
View
EC50
-
=
0.007
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009171
PGDB_C008792
PGDB_AS001244
View
EC50
-
=
0.136
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009249
PGDB_C008870
PGDB_AS001244
View
EC50
-
=
0.017
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009400
PGDB_C008848
PGDB_AS001244
View
EC50
-
=
0.13
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A009467
PGDB_C008865
PGDB_AS001244
View
EC50
-
=
0.048
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A010331
PGDB_C008810
PGDB_AS001244
View
EC50
-
=
0.411
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A010654
PGDB_C008897
PGDB_AS001244
View
EC50
-
=
0.012
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A010775
PGDB_C008819
PGDB_AS001244
View
EC50
-
=
0.014
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A010996
PGDB_C008823
PGDB_AS001244
View
EC50
-
=
0.006
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011379
PGDB_C008845
PGDB_AS001244
View
EC50
-
=
0.11
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011445
PGDB_C008931
PGDB_AS001244
View
EC50
-
=
0.009
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011567
PGDB_C008837
PGDB_AS001244
View
EC50
-
=
0.88
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011598
PGDB_C008874
PGDB_AS001244
View
EC50
-
=
1.31
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011679
PGDB_C008920
PGDB_AS001244
View
EC50
-
=
0.037
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011723
PGDB_C008761
PGDB_AS001244
View
EC50
-
=
0.007
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A011957
PGDB_C008853
PGDB_AS001244
View
EC50
-
=
0.082
mM
-
—
IKZF2
-
293GT
KR20210031680A
PGDB_A013648
PGDB_C008911
PGDB_AS001244
View