Assay
PGDB_AS001269
System: cell_basedCell line: MDA-MB-231
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 5 | nM | - | — | - | - | MDA-MB-231 | WO2024032689A1 | PGDB_A027072 | PGDB_C002489 | PGDB_AS001269 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | MDA-MB-231 | WO2024032689A1 | PGDB_A033013 | PGDB_C002488 | PGDB_AS001269 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MDA-MB-231 | WO2024032689A1 | PGDB_A052140 | PGDB_C002490 | PGDB_AS001269 | View | |
| IC50 | - | = | 50-100 | nM | - | — | - | - | MDA-MB-231 | WO2024032689A1 | PGDB_A065707 | PGDB_C002487 | PGDB_AS001269 | View | |
| IC50 | - | <= | 5 | nM | - | — | - | - | MDA-MB-231 | WO2024032689A1 | PGDB_A073389 | PGDB_C002491 | PGDB_AS001269 | View |