Assay
PGDB_AS001451
System: cell_basedTarget: CRBN | DDB1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 97.43 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A008908 | PGDB_C007379 | PGDB_AS001451 | View | |
| % Inhibition | - | = | 98.81 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A023228 | PGDB_C007378 | PGDB_AS001451 | View | |
| % Inhibition | - | = | 98.91 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A035859 | PGDB_C007375 | PGDB_AS001451 | View | |
| % Inhibition | - | = | 100.05 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A050296 | PGDB_C007374 | PGDB_AS001451 | View | |
| % Inhibition | - | = | 98.34 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A065379 | PGDB_C007376 | PGDB_AS001451 | View | |
| % Inhibition | - | = | 97.86 | % | Concentration series: 50 uM, 100 uM | 2 h | CRBN | CRBN | - | CN121378270A | PGDB_A065430 | PGDB_C007377 | PGDB_AS001451 | View |