Assay
PGDB_AS001461
System: cell_basedCell line: FaDu
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 205.4 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A012808 | PGDB_C006026 | PGDB_AS001461 | View | |
| IC50 | - | = | 1.528 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A017359 | PGDB_C006025 | PGDB_AS001461 | View | |
| IC50 | - | = | 73.24 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A019714 | PGDB_C006028 | PGDB_AS001461 | View | |
| IC50 | - | = | 3.369 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A024985 | PGDB_C006028 | PGDB_AS001461 | View | |
| IC50 | - | = | 109 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A029927 | PGDB_C006027 | PGDB_AS001461 | View | |
| IC50 | - | = | 22.51 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A049733 | PGDB_C006025 | PGDB_AS001461 | View | |
| IC50 | - | = | 7.022 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A051632 | PGDB_C006027 | PGDB_AS001461 | View | |
| IC50 | - | = | 7.46 | nM | - | — | DDX5 | - | FaDu | AU2023256446A1 | PGDB_A072518 | PGDB_C006026 | PGDB_AS001461 | View |