Assay context summary

Assay context

81 activity records
Activity compounds and values

Activity records

81 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007106
IC50-=9.7nM-PDE3A-SK-MEL-3CN120265631APGDB_A007655PGDB_C007106PGDB_AS001659View
2D structure for PGDB_C007104
IC50-=0.4nM-PDE3A-SK-MEL-3CN120265631APGDB_A007838PGDB_C007104PGDB_AS001659View
2D structure for PGDB_C007087
IC50-=1.6nM-PDE3A-SK-MEL-3CN120265631APGDB_A008379PGDB_C007087PGDB_AS001659View
2D structure for PGDB_C007144
IC50-=5.2nM-PDE3A-SK-MEL-3CN120265631APGDB_A009197PGDB_C007144PGDB_AS001659View
2D structure for PGDB_C007107
IC50-=4.4nM-PDE3A-SK-MEL-3CN120265631APGDB_A010257PGDB_C007107PGDB_AS001659View
2D structure for PGDB_C007095
IC50-=2.3nM-PDE3A-SK-MEL-3CN120265631APGDB_A010687PGDB_C007095PGDB_AS001659View
2D structure for PGDB_C007093
IC50-=1.6nM-PDE3A-SK-MEL-3CN120265631APGDB_A010688PGDB_C007093PGDB_AS001659View
2D structure for PGDB_C007140
IC50-=0.07nM-PDE3A-SK-MEL-3CN120265631APGDB_A011374PGDB_C007140PGDB_AS001659View
2D structure for PGDB_C007082
IC50-=0.8nM-PDE3A-SK-MEL-3CN120265631APGDB_A011933PGDB_C007082PGDB_AS001659View
2D structure for PGDB_C007115
IC50-=2.5nM-PDE3A-SK-MEL-3CN120265631APGDB_A012926PGDB_C007115PGDB_AS001659View
2D structure for PGDB_C007112
IC50-=1.1nM-PDE3A-SK-MEL-3CN120265631APGDB_A013410PGDB_C007112PGDB_AS001659View
2D structure for PGDB_C007070
IC50-=0.4nM-PDE3A-SK-MEL-3CN120265631APGDB_A013584PGDB_C007070PGDB_AS001659View
2D structure for PGDB_C007110
IC50-=74.6nM-PDE3A-SK-MEL-3CN120265631APGDB_A013849PGDB_C007110PGDB_AS001659View
2D structure for PGDB_C007074
IC50-=4.1nM-PDE3A-SK-MEL-3CN120265631APGDB_A015614PGDB_C007074PGDB_AS001659View
2D structure for PGDB_C007119
IC50-=0.9nM-PDE3A-SK-MEL-3CN120265631APGDB_A015822PGDB_C007119PGDB_AS001659View
2D structure for PGDB_C007156
IC50-=258.1nM-PDE3A-SK-MEL-3CN120265631APGDB_A017272PGDB_C007156PGDB_AS001659View
2D structure for PGDB_C007086
IC50-=0.7nM-PDE3A-SK-MEL-3CN120265631APGDB_A017589PGDB_C007086PGDB_AS001659View
2D structure for PGDB_C007072
IC50-=1.2nM-PDE3A-SK-MEL-3CN120265631APGDB_A018458PGDB_C007072PGDB_AS001659View
2D structure for PGDB_C007147
IC50-=0.3nM-PDE3A-SK-MEL-3CN120265631APGDB_A018589PGDB_C007147PGDB_AS001659View
2D structure for PGDB_C007065
IC50-=37.9nM-PDE3A-SK-MEL-3CN120265631APGDB_A018988PGDB_C007065PGDB_AS001659View