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SIMM · NJU
Assay
PGDB_AS001674
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
136 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
136 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
6
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A007211
PGDB_C011282
PGDB_AS001674
View
Dmax
-
=
7.5
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A007583
PGDB_C011364
PGDB_AS001674
View
Dmax
-
=
2.9
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A007946
PGDB_C011339
PGDB_AS001674
View
Dmax
-
=
2.6
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A009498
PGDB_C011371
PGDB_AS001674
View
Dmax
-
=
5.1
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A009631
PGDB_C011288
PGDB_AS001674
View
Dmax
-
=
14.6
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A010014
PGDB_C011314
PGDB_AS001674
View
Dmax
-
=
6.9
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A010729
PGDB_C011349
PGDB_AS001674
View
Dmax
-
=
12.1
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A012037
PGDB_C011309
PGDB_AS001674
View
Dmax
-
=
13.6
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A015264
PGDB_C011385
PGDB_AS001674
View
Dmax
-
=
11.4
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A015427
PGDB_C011329
PGDB_AS001674
View
Dmax
-
=
5.9
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A015884
PGDB_C011354
PGDB_AS001674
View
Dmax
-
=
8.4
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A016150
PGDB_C011312
PGDB_AS001674
View
Dmax
-
=
18.4
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A016485
PGDB_C011346
PGDB_AS001674
View
Dmax
-
=
7.6
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A017138
PGDB_C011381
PGDB_AS001674
View
Dmax
-
=
10.3
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A017404
PGDB_C011391
PGDB_AS001674
View
Dmax
-
=
5.4
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A017568
PGDB_C011324
PGDB_AS001674
View
Dmax
-
=
12.2
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A018193
PGDB_C011325
PGDB_AS001674
View
Dmax
-
=
10.2
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A018425
PGDB_C011297
PGDB_AS001674
View
Dmax
-
=
3
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A018587
PGDB_C011331
PGDB_AS001674
View
Dmax
-
=
5.1
%
-
-
GSPT1
-
HEK293
WO2025181261A1
PGDB_A021113
PGDB_C011341
PGDB_AS001674
View