Assay context summary

Assay context

320 activity records
Activity compounds and values

Activity records

320 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020732
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007029PGDB_C020732PGDB_AS001676View
2D structure for PGDB_C020605
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007328PGDB_C020605PGDB_AS001676View
2D structure for PGDB_C020721
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007733PGDB_C020721PGDB_AS001676View
2D structure for PGDB_C020682
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007779PGDB_C020682PGDB_AS001676View
2D structure for PGDB_C020530
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007803PGDB_C020530PGDB_AS001676View
2D structure for PGDB_C020684
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007804PGDB_C020684PGDB_AS001676View
2D structure for PGDB_C020538
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007831PGDB_C020538PGDB_AS001676View
2D structure for PGDB_C020693
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008034PGDB_C020693PGDB_AS001676View
2D structure for PGDB_C020741
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008073PGDB_C020741PGDB_AS001676View
2D structure for PGDB_C020554
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008292PGDB_C020554PGDB_AS001676View
2D structure for PGDB_C020771
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008331PGDB_C020771PGDB_AS001676View
2D structure for PGDB_C020521
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008445PGDB_C020521PGDB_AS001676View
2D structure for PGDB_C020585
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008788PGDB_C020585PGDB_AS001676View
2D structure for PGDB_C020665
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008887PGDB_C020665PGDB_AS001676View
2D structure for PGDB_C020495
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009319PGDB_C020495PGDB_AS001676View
2D structure for PGDB_C020618
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009372PGDB_C020618PGDB_AS001676View
2D structure for PGDB_C020675
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009429PGDB_C020675PGDB_AS001676View
2D structure for PGDB_C020625
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009509PGDB_C020625PGDB_AS001676View
2D structure for PGDB_C020645
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009643PGDB_C020645PGDB_AS001676View
2D structure for PGDB_C020634
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A009815PGDB_C020634PGDB_AS001676View