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SIMM · NJU
Assay
PGDB_AS001690
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
58 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
GSPT1
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
58 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000098
PGDB_C031976
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000359
PGDB_C031995
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000467
PGDB_C031943
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000626
PGDB_C031993
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000705
PGDB_C031984
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A000860
PGDB_C031946
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001013
PGDB_C031976
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001207
PGDB_C031989
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001506
PGDB_C031973
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001509
PGDB_C031959
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001559
PGDB_C031974
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A001711
PGDB_C031954
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002037
PGDB_C031975
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002153
PGDB_C031953
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002506
PGDB_C031968
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002530
PGDB_C031988
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002599
PGDB_C031952
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002687
PGDB_C031969
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A002773
PGDB_C031950
PGDB_AS001690
View
DC50
-
>
3000
nM
-
—
GSPT1
CRBN
HEK293
WO2026114958A1
PGDB_A003210
PGDB_C031964
PGDB_AS001690
View