Assay
PGDB_AS001722
System: cell_basedTarget: CUL4BCell line: KBM7
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| LC50 | - | = | 5.682 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A007968 | PGDB_C019080 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A028350 | PGDB_C019071 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A032137 | PGDB_C019074 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A040711 | PGDB_C019073 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A043989 | PGDB_C019078 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A056056 | PGDB_C019077 | PGDB_AS001722 | View | |
| LC50 | - | = | 6.061 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A059140 | PGDB_C019075 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A067317 | PGDB_C019081 | PGDB_AS001722 | View | |
| LC50 | - | = | 2.005 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A072654 | PGDB_C019079 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A074421 | PGDB_C019076 | PGDB_AS001722 | View | |
| LC50 | - | > | 10 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A075350 | PGDB_C019072 | PGDB_AS001722 | View |