Assay
PGDB_AS001753
System: cell_basedTarget: IKZF2Cell line: HEK293T
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.005 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A009740 | PGDB_C000388 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.292 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A016828 | PGDB_C000384 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.024 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A021733 | PGDB_C000380 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.0005 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A036021 | PGDB_C000389 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A040990 | PGDB_C000386 | PGDB_AS001753 | View | |
| DC50 | - | > | 30 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A046347 | PGDB_C000382 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.005 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A056586 | PGDB_C000387 | PGDB_AS001753 | View | |
| DC50 | - | > | 30 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A060685 | PGDB_C000383 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A069678 | PGDB_C000385 | PGDB_AS001753 | View | |
| DC50 | - | = | 0.006 | uM | - | — | IKZF2 | - | HEK293T | AR126418A1 | PGDB_A072203 | PGDB_C000381 | PGDB_AS001753 | View |