Assay
PGDB_AS001757
System: cell_basedTarget: VAV1Cell line: Jurkat
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 90.405 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A008979 | PGDB_C009238 | PGDB_AS001757 | View | |
| Dmax | - | = | 86.33 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A010929 | PGDB_C009199 | PGDB_AS001757 | View | |
| Dmax | - | = | 83.377 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A011659 | PGDB_C009203 | PGDB_AS001757 | View | |
| Dmax | - | = | 70.243 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A012740 | PGDB_C009241 | PGDB_AS001757 | View | |
| Dmax | - | = | 94.146 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A013466 | PGDB_C009181 | PGDB_AS001757 | View | |
| Dmax | - | = | 91.307 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A014630 | PGDB_C009189 | PGDB_AS001757 | View | |
| Dmax | - | = | 66.69 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A016715 | PGDB_C009216 | PGDB_AS001757 | View | |
| Dmax | - | = | 95.443 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A017417 | PGDB_C009176 | PGDB_AS001757 | View | |
| Dmax | - | = | 94.916 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A017716 | PGDB_C009178 | PGDB_AS001757 | View | |
| Dmax | - | = | 93.791 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A018239 | PGDB_C009237 | PGDB_AS001757 | View | |
| Dmax | - | = | 83.574 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A018516 | PGDB_C009202 | PGDB_AS001757 | View | |
| Dmax | - | = | 92.999 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A018628 | PGDB_C009185 | PGDB_AS001757 | View | |
| Dmax | - | = | 97.919 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A018758 | PGDB_C009168 | PGDB_AS001757 | View | |
| Dmax | - | = | 91.031 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A019814 | PGDB_C009234 | PGDB_AS001757 | View | |
| Dmax | - | = | 78.314 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A020002 | PGDB_C009208 | PGDB_AS001757 | View | |
| Dmax | - | = | 90.47 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A020177 | PGDB_C009194 | PGDB_AS001757 | View | |
| Dmax | - | = | 53.134 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A021486 | PGDB_C009225 | PGDB_AS001757 | View | |
| Dmax | - | = | 78.312 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A021622 | PGDB_C009209 | PGDB_AS001757 | View | |
| Dmax | - | = | 37.533 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A021849 | PGDB_C009230 | PGDB_AS001757 | View | |
| Dmax | - | = | 92.863 | % | Concentration series: 10 uM, 0.5 nM | 24 h | VAV1 | - | Jurkat | WO2026013576A1 | PGDB_A022317 | PGDB_C009187 | PGDB_AS001757 | View |