Assay context summary

Assay context

77 activity records
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C009238
Dmax-=90.405%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A008979PGDB_C009238PGDB_AS001757View
2D structure for PGDB_C009199
Dmax-=86.33%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A010929PGDB_C009199PGDB_AS001757View
2D structure for PGDB_C009203
Dmax-=83.377%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A011659PGDB_C009203PGDB_AS001757View
2D structure for PGDB_C009241
Dmax-=70.243%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A012740PGDB_C009241PGDB_AS001757View
2D structure for PGDB_C009181
Dmax-=94.146%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A013466PGDB_C009181PGDB_AS001757View
2D structure for PGDB_C009189
Dmax-=91.307%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A014630PGDB_C009189PGDB_AS001757View
2D structure for PGDB_C009216
Dmax-=66.69%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A016715PGDB_C009216PGDB_AS001757View
2D structure for PGDB_C009176
Dmax-=95.443%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A017417PGDB_C009176PGDB_AS001757View
2D structure for PGDB_C009178
Dmax-=94.916%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A017716PGDB_C009178PGDB_AS001757View
2D structure for PGDB_C009237
Dmax-=93.791%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A018239PGDB_C009237PGDB_AS001757View
2D structure for PGDB_C009202
Dmax-=83.574%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A018516PGDB_C009202PGDB_AS001757View
2D structure for PGDB_C009185
Dmax-=92.999%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A018628PGDB_C009185PGDB_AS001757View
2D structure for PGDB_C009168
Dmax-=97.919%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A018758PGDB_C009168PGDB_AS001757View
2D structure for PGDB_C009234
Dmax-=91.031%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A019814PGDB_C009234PGDB_AS001757View
2D structure for PGDB_C009208
Dmax-=78.314%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A020002PGDB_C009208PGDB_AS001757View
2D structure for PGDB_C009194
Dmax-=90.47%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A020177PGDB_C009194PGDB_AS001757View
2D structure for PGDB_C009225
Dmax-=53.134%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A021486PGDB_C009225PGDB_AS001757View
2D structure for PGDB_C009209
Dmax-=78.312%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A021622PGDB_C009209PGDB_AS001757View
2D structure for PGDB_C009230
Dmax-=37.533%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A021849PGDB_C009230PGDB_AS001757View
2D structure for PGDB_C009187
Dmax-=92.863%Concentration series: 10 uM, 0.5 nM24 hVAV1-JurkatWO2026013576A1PGDB_A022317PGDB_C009187PGDB_AS001757View