Assay

PGDB_AS001844

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

114 activity records
Assay familybiochemical
Systembiochemical
ReadoutKi
TargetCRBN | DDB1
E3CRBN | DDB1
Organismrecombinant protein system
TechnologyHTRF
Activity compounds and values

Activity records

114 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C027487
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A008432PGDB_C027487PGDB_AS001844View
2D structure for PGDB_C027491
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A009003PGDB_C027491PGDB_AS001844View
2D structure for PGDB_C027570
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A009443PGDB_C027570PGDB_AS001844View
2D structure for PGDB_C027480
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A010461PGDB_C027480PGDB_AS001844View
2D structure for PGDB_C027558
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A010661PGDB_C027558PGDB_AS001844View
2D structure for PGDB_C027554
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A011400PGDB_C027554PGDB_AS001844View
2D structure for PGDB_C027488
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A012036PGDB_C027488PGDB_AS001844View
2D structure for PGDB_C027495
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A012436PGDB_C027495PGDB_AS001844View
2D structure for PGDB_C027517
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A012770PGDB_C027517PGDB_AS001844View
2D structure for PGDB_C027576
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A012975PGDB_C027576PGDB_AS001844View
2D structure for PGDB_C027528
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A013009PGDB_C027528PGDB_AS001844View
2D structure for PGDB_C027468
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A015029PGDB_C027468PGDB_AS001844View
2D structure for PGDB_C027506
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A015512PGDB_C027506PGDB_AS001844View
2D structure for PGDB_C027525
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A016000PGDB_C027525PGDB_AS001844View
2D structure for PGDB_C027572
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A016543PGDB_C027572PGDB_AS001844View
2D structure for PGDB_C027530
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A016704PGDB_C027530PGDB_AS001844View
2D structure for PGDB_C027512
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A016892PGDB_C027512PGDB_AS001844View
2D structure for PGDB_C027562
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A018153PGDB_C027562PGDB_AS001844View
2D structure for PGDB_C027493
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A018210PGDB_C027493PGDB_AS001844View
2D structure for PGDB_C027518
Ki-<=0.1uM-—CRBNCRBN-WO2025224262A1PGDB_A020222PGDB_C027518PGDB_AS001844View
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