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SIMM · NJU
Assay
PGDB_AS001862
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
733 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
GSPT1
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
733 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007019
PGDB_C003929
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007214
PGDB_C003698
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007229
PGDB_C003635
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007267
PGDB_C003584
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007361
PGDB_C003494
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007630
PGDB_C003525
PGDB_AS001862
View
DC50
-
<
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007750
PGDB_C003928
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007787
PGDB_C004053
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007910
PGDB_C003666
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007965
PGDB_C003959
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A007984
PGDB_C003778
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008050
PGDB_C003543
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008058
PGDB_C003886
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008127
PGDB_C003716
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008270
PGDB_C003977
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008536
PGDB_C003820
PGDB_AS001862
View
DC50
-
<
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008584
PGDB_C003849
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008600
PGDB_C003975
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008629
PGDB_C004079
PGDB_AS001862
View
DC50
-
>=
25
nM
-
—
GSPT1
-
HEK293
EP4584259A1
PGDB_A008694
PGDB_C003490
PGDB_AS001862
View