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SIMM · NJU
Assay
PGDB_AS001899
System: biochemical
Target: CRBN
Assay context summary
Assay context
115 activity records
Assay family
biochemical
System
biochemical
Readout
Ki
Target
CRBN
E3
CRBN
Organism
recombinant protein system
Technology
HTRF
Activity compounds and values
Activity records
115 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A007743
PGDB_C027568
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A008773
PGDB_C027571
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A009076
PGDB_C027453
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A009092
PGDB_C027461
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A009690
PGDB_C027506
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A009897
PGDB_C027502
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A010067
PGDB_C027469
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A010360
PGDB_C027577
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A010794
PGDB_C027466
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A011037
PGDB_C027515
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A011052
PGDB_C027553
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A011370
PGDB_C027524
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A012574
PGDB_C027521
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A013743
PGDB_C027467
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A013844
PGDB_C027511
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A013876
PGDB_C027556
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A013985
PGDB_C027517
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A015216
PGDB_C027472
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A015894
PGDB_C027564
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
WO2024092039
PGDB_A016062
PGDB_C027455
PGDB_AS001899
View