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SIMM · NJU
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SIMM · NJU
Patent
WO2024092039
128 compounds
160 activity records
2 assays
Patent summary
Publication number
WO2024092039
Assignee
Monte Rosa Therapeutics
Family members
2
Family patent IDs
CL2025001171A1
WO2024092039A1
Filing year
2,023
Jurisdiction
WO
Compounds
128
Activity records
160
Assays
2
Activity compounds and values
Activity records
160 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A007194
PGDB_C027513
PGDB_AS002575
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A007743
PGDB_C027568
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A008773
PGDB_C027571
PGDB_AS001899
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A008837
PGDB_C027499
PGDB_AS002575
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A009076
PGDB_C027453
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A009092
PGDB_C027461
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A009690
PGDB_C027506
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A009897
PGDB_C027502
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A010067
PGDB_C027469
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A010360
PGDB_C027577
PGDB_AS001899
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A010580
PGDB_C027547
PGDB_AS002575
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A010794
PGDB_C027466
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A011037
PGDB_C027515
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A011052
PGDB_C027553
PGDB_AS001899
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A011328
PGDB_C027461
PGDB_AS002575
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A011370
PGDB_C027524
PGDB_AS001899
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A012574
PGDB_C027521
PGDB_AS001899
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A012934
PGDB_C027500
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
PGDB_A013709
PGDB_C027535
PGDB_AS002575
View
Ki
-
<=
0.1
uM
-
—
-
-
-
PGDB_A013743
PGDB_C027467
PGDB_AS001899
View