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SIMM · NJU
Assay
PGDB_AS002080
System: biochemical
Target: NFE2L2
Assay context summary
Assay context
198 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
NFE2L2
E3
BTRC | FBXW11 | SKP1
Activity compounds and values
Activity records
198 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007219
PGDB_C020796
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007571
PGDB_C020816
PGDB_AS002080
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007685
PGDB_C020830
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A008781
PGDB_C020894
PGDB_AS002080
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009142
PGDB_C020907
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009672
PGDB_C020826
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009910
PGDB_C020965
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010297
PGDB_C020812
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010355
PGDB_C020954
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A011686
PGDB_C020944
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013012
PGDB_C020963
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013265
PGDB_C020855
PGDB_AS002080
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A014048
PGDB_C020849
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015062
PGDB_C020945
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015196
PGDB_C020890
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015215
PGDB_C020838
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015519
PGDB_C020937
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A017103
PGDB_C020795
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A017106
PGDB_C020833
PGDB_AS002080
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
WO2025179005A1
PGDB_A017685
PGDB_C020874
PGDB_AS002080
View