Assay
PGDB_AS002106
System: cell_basedCell line: KBM7
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| LC50 | - | = | 6.993 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A013585 | PGDB_C019080 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A018297 | PGDB_C019076 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A021539 | PGDB_C019077 | PGDB_AS002106 | View | |
| LC50 | - | = | 2.748 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A026507 | PGDB_C019079 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A031797 | PGDB_C019078 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A045229 | PGDB_C019072 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A048971 | PGDB_C019081 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A050593 | PGDB_C019073 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A053730 | PGDB_C019074 | PGDB_AS002106 | View | |
| LC50 | - | > | 10 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A068554 | PGDB_C019071 | PGDB_AS002106 | View | |
| LC50 | - | = | 6.797 | uM | - | — | CCNK | - | KBM7 | AU2021359129A1 | PGDB_A071749 | PGDB_C019075 | PGDB_AS002106 | View |