Assay
PGDB_AS002207
System: cell_basedCell line: NCI-N87
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A010786 | PGDB_C001022 | PGDB_AS002207 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A014830 | PGDB_C001023 | PGDB_AS002207 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A021298 | PGDB_C001025 | PGDB_AS002207 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A031605 | PGDB_C001020 | PGDB_AS002207 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A032425 | PGDB_C001026 | PGDB_AS002207 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A035558 | PGDB_C001019 | PGDB_AS002207 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A052224 | PGDB_C001018 | PGDB_AS002207 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A056274 | PGDB_C001027 | PGDB_AS002207 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A072863 | PGDB_C001024 | PGDB_AS002207 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | NCI-N87 | CN121219280A | PGDB_A074770 | PGDB_C001021 | PGDB_AS002207 | View |