PatGlueDB | Molecular Glue Patent Bioactivity Database

Assay context summary

Assay context

83 activity records

Assay family% Degradation

Systemcell_based

ReadoutDC50

TargetGSPT1

E3CRBN

Cell lineCAL-51

OrganismHomo sapiens

Technologyfluorescence

Activity compounds and values

Activity records

83 records

Metric	Control	Relation	Value	Unit	Concentration	Time	Target	E3	Cell line	Patent	Record ID	Compound	Assay	Details
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A007453	PGDB_C021949	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A009067	PGDB_C021954	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A009599	PGDB_C021937	PGDB_AS002250	View
DC50	-	<=	30	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A011413	PGDB_C000378	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A012055	PGDB_C021958	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A012110	PGDB_C021944	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A013337	PGDB_C021972	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A013537	PGDB_C021916	PGDB_AS002250	View
DC50	-	<=	30	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A014175	PGDB_C021965	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A016365	PGDB_C021906	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A017194	PGDB_C021902	PGDB_AS002250	View
DC50	-	<=	30	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A018385	PGDB_C021914	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A018963	PGDB_C021904	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A019198	PGDB_C021912	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A020168	PGDB_C021896	PGDB_AS002250	View
DC50	-	<=	30	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A020361	PGDB_C021974	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A021041	PGDB_C021946	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A022020	PGDB_C021939	PGDB_AS002250	View
DC50	-	>	300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A022842	PGDB_C021908	PGDB_AS002250	View
DC50	-	=	30-300	nM	-	—	-	-	CAL-51	AU2022207648A1	PGDB_A023827	PGDB_C021959	PGDB_AS002250	View

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