Assay context summary

Assay context

58 activity records
Activity compounds and values

Activity records

58 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031977
IC50-=2.2nM--CRBNSK-CO-1WO2026114958A1PGDB_A000269PGDB_C031977PGDB_AS002392View
2D structure for PGDB_C031978
IC50-=1.7nM--CRBNSK-CO-1WO2026114958A1PGDB_A000434PGDB_C031978PGDB_AS002392View
2D structure for PGDB_C031985
IC50-=0.8nM--CRBNSK-CO-1WO2026114958A1PGDB_A000765PGDB_C031985PGDB_AS002392View
2D structure for PGDB_C031967
IC50-=4.6nM--CRBNSK-CO-1WO2026114958A1PGDB_A001106PGDB_C031967PGDB_AS002392View
2D structure for PGDB_C031976
IC50-=4.5nM--CRBNSK-CO-1WO2026114958A1PGDB_A001203PGDB_C031976PGDB_AS002392View
2D structure for PGDB_C031970
IC50-=2.4nM--CRBNSK-CO-1WO2026114958A1PGDB_A001446PGDB_C031970PGDB_AS002392View
2D structure for PGDB_C031943
IC50-=4.5nM--CRBNSK-CO-1WO2026114958A1PGDB_A001590PGDB_C031943PGDB_AS002392View
2D structure for PGDB_C031990
IC50-=2.1nM--CRBNSK-CO-1WO2026114958A1PGDB_A001832PGDB_C031990PGDB_AS002392View
2D structure for PGDB_C031976
IC50-=7.8nM--CRBNSK-CO-1WO2026114958A1PGDB_A001846PGDB_C031976PGDB_AS002392View
2D structure for PGDB_C031942
IC50-=1.4nM--CRBNSK-CO-1WO2026114958A1PGDB_A001893PGDB_C031942PGDB_AS002392View
2D structure for PGDB_C031995
IC50-=1.2nM--CRBNSK-CO-1WO2026114958A1PGDB_A002137PGDB_C031995PGDB_AS002392View
2D structure for PGDB_C031988
IC50-=8.4nM--CRBNSK-CO-1WO2026114958A1PGDB_A002242PGDB_C031988PGDB_AS002392View
2D structure for PGDB_C031962
IC50-=1.3nM--CRBNSK-CO-1WO2026114958A1PGDB_A002320PGDB_C031962PGDB_AS002392View
2D structure for PGDB_C031957
IC50-=4.1nM--CRBNSK-CO-1WO2026114958A1PGDB_A002386PGDB_C031957PGDB_AS002392View
2D structure for PGDB_C031968
IC50-=0.8nM--CRBNSK-CO-1WO2026114958A1PGDB_A002550PGDB_C031968PGDB_AS002392View
2D structure for PGDB_C031994
IC50-=1.7nM--CRBNSK-CO-1WO2026114958A1PGDB_A002625PGDB_C031994PGDB_AS002392View
2D structure for PGDB_C031964
IC50-=8.1nM--CRBNSK-CO-1WO2026114958A1PGDB_A002683PGDB_C031964PGDB_AS002392View
2D structure for PGDB_C031981
IC50-=6.5nM--CRBNSK-CO-1WO2026114958A1PGDB_A003095PGDB_C031981PGDB_AS002392View
2D structure for PGDB_C031971
IC50-=1nM--CRBNSK-CO-1WO2026114958A1PGDB_A003208PGDB_C031971PGDB_AS002392View
2D structure for PGDB_C031989
IC50-=4.8nM--CRBNSK-CO-1WO2026114958A1PGDB_A003310PGDB_C031989PGDB_AS002392View