Assay
PGDB_AS002507
System: cell_basedCell line: KBM7
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| LC50 | - | = | 1.812 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A008354 | PGDB_C019076 | PGDB_AS002507 | View | |
| LC50 | - | = | 7.121 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A029418 | PGDB_C019071 | PGDB_AS002507 | View | |
| LC50 | - | = | 2.352 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A030786 | PGDB_C019077 | PGDB_AS002507 | View | |
| LC50 | - | = | 7.821 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A040898 | PGDB_C019078 | PGDB_AS002507 | View | |
| LC50 | - | = | 4.693 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A058422 | PGDB_C019081 | PGDB_AS002507 | View | |
| LC50 | - | = | 3.747 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A063304 | PGDB_C019074 | PGDB_AS002507 | View | |
| LC50 | - | = | 0.92 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A070583 | PGDB_C019079 | PGDB_AS002507 | View | |
| LC50 | - | = | 1.35 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A072837 | PGDB_C019072 | PGDB_AS002507 | View | |
| LC50 | - | = | 1.286 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A073676 | PGDB_C019080 | PGDB_AS002507 | View | |
| LC50 | - | = | 1.569 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A075681 | PGDB_C019075 | PGDB_AS002507 | View | |
| LC50 | - | = | 11.75 | uM | - | — | - | - | KBM7 | AU2021359129A1 | PGDB_A077162 | PGDB_C019073 | PGDB_AS002507 | View |