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SIMM · NJU
Assay
PGDB_AS002572
System: cell_based
Target: NEK7
Cell line: CAL-51
Assay context summary
Assay context
93 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
NEK7
E3
CRBN
Cell line
CAL-51
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
93 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A008620
PGDB_C026263
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A008707
PGDB_C026256
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A009316
PGDB_C020248
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A010534
PGDB_C020212
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A010801
PGDB_C020213
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A011456
PGDB_C026233
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A011564
PGDB_C026274
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A011728
PGDB_C026264
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A013574
PGDB_C026241
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014362
PGDB_C026248
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014402
PGDB_C020245
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014407
PGDB_C020179
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014913
PGDB_C026238
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A014930
PGDB_C020200
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A016147
PGDB_C026271
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A016217
PGDB_C020247
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A016261
PGDB_C020195
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A016990
PGDB_C026255
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A017989
PGDB_C026265
PGDB_AS002572
View
DC50
-
<=
100
nM
-
—
-
-
CAL-51
KR20260041885A
PGDB_A018370
PGDB_C020214
PGDB_AS002572
View