Summary
AssigneeInstitute of Medicinal Biotechnology, CAMS & PUMC
Filing years2022
Patents1
Compounds15
Activity records44
Patent families1
Targets1
Assay familiescellular_function, degradation, viability
Activity metricsCC50, EC50
Overview

Target distribution and active-compound trend

Target distribution

44 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

08152024
Activity compounds and values

Activity records

44 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C008304
EC50-=27.85uM-BLOC1S6-HEK293TJP2024545831APGDB_A008434PGDB_C008304PGDB_AS002050View
2D structure for PGDB_C008307
EC50-=0.88uM-BLOC1S6-HEK293TJP2024545831APGDB_A008589PGDB_C008307PGDB_AS002145View
2D structure for PGDB_C008299
EC50-=1.14uM-BLOC1S6-HEK293TJP2024545831APGDB_A014449PGDB_C008299PGDB_AS002145View
2D structure for PGDB_C008306
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A014802PGDB_C008306PGDB_AS001447View
2D structure for PGDB_C008307
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A016530PGDB_C008307PGDB_AS001447View
2D structure for PGDB_C008298
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A018938PGDB_C008298PGDB_AS001447View
2D structure for PGDB_C008302
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A019225PGDB_C008302PGDB_AS001447View
2D structure for PGDB_C008309
EC50-=0.92uM-BLOC1S6-HEK293TJP2024545831APGDB_A019604PGDB_C008309PGDB_AS002050View
2D structure for PGDB_C008307
EC50-=1.22uM-BLOC1S6-HEK293TJP2024545831APGDB_A021762PGDB_C008307PGDB_AS002050View
2D structure for PGDB_C008311
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A021887PGDB_C008311PGDB_AS001447View
2D structure for PGDB_C008305
EC50-=0.55uM-BLOC1S6-HEK293TJP2024545831APGDB_A024237PGDB_C008305PGDB_AS002050View
2D structure for PGDB_C008302
EC50-=2.09uM-BLOC1S6-HEK293TJP2024545831APGDB_A024374PGDB_C008302PGDB_AS002145View
2D structure for PGDB_C008309
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A025667PGDB_C008309PGDB_AS001447View
2D structure for PGDB_C008302
EC50-=2.22uM-BLOC1S6-HEK293TJP2024545831APGDB_A027459PGDB_C008302PGDB_AS002050View
2D structure for PGDB_C008298
EC50-=0.58uM-BLOC1S6-HEK293TJP2024545831APGDB_A028847PGDB_C008298PGDB_AS002050View
2D structure for PGDB_C008301
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A029126PGDB_C008301PGDB_AS001447View
2D structure for PGDB_C008300
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A033885PGDB_C008300PGDB_AS001447View
2D structure for PGDB_C008305
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A034299PGDB_C008305PGDB_AS001447View
2D structure for PGDB_C008300
EC50-=1.25uM-BLOC1S6-HEK293TJP2024545831APGDB_A035574PGDB_C008300PGDB_AS002050View
2D structure for PGDB_C008308
CC50->100uM-BLOC1S6-HEK293TJP2024545831APGDB_A037590PGDB_C008308PGDB_AS001447View