Summary
AssigneeKorea Research Institute Of Bioscience And Biotechnology Kribb
Filing years2024
Patents1
Compounds114
Activity records128
Patent families1
Targets1
Assay familiesdegradation
Activity metricsdegradation
Overview

Target distribution and active-compound trend

Target distribution

253 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0561122025
Activity compounds and values

Activity records

253 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C025442
% Degradation-=6.4%----JurkatEP4660193A1PGDB_A007020PGDB_C025442PGDB_AS000451View
2D structure for PGDB_C025421
% Degradation-=50.9%--IKZF2-JurkatEP4660193A1PGDB_A007121PGDB_C025421PGDB_AS002037View
2D structure for PGDB_C025483
% Degradation-=21.3%--IKZF2-JurkatEP4660193A1PGDB_A007149PGDB_C025483PGDB_AS002037View
2D structure for PGDB_C025506
% Degradation-=89.1%----JurkatEP4660193A1PGDB_A007151PGDB_C025506PGDB_AS000451View
2D structure for PGDB_C025476
% Degradation-=94.6%--IKZF2-JurkatEP4660193A1PGDB_A007477PGDB_C025476PGDB_AS002037View
2D structure for PGDB_C025525
DC50-<10.0nM---JurkatEP4660193A1PGDB_A007668PGDB_C025525PGDB_AS001105View
2D structure for PGDB_C025422
% Degradation-=21.7%----JurkatEP4660193A1PGDB_A007879PGDB_C025422PGDB_AS000451View
2D structure for PGDB_C025524
Dmax-=100.0%----JurkatEP4660193A1PGDB_A007927PGDB_C025524PGDB_AS000303View
2D structure for PGDB_C025502
Dmax-=100.0%----JurkatEP4660193A1PGDB_A008345PGDB_C025502PGDB_AS000303View
2D structure for PGDB_C025523
Dmax-=96.0%----JurkatEP4660193A1PGDB_A008468PGDB_C025523PGDB_AS000303View
2D structure for PGDB_C025449
% Degradation-=28.7%----JurkatEP4660193A1PGDB_A009032PGDB_C025449PGDB_AS000451View
2D structure for PGDB_C025441
% Degradation-=11.8%--IKZF2-JurkatEP4660193A1PGDB_A009405PGDB_C025441PGDB_AS002037View
2D structure for PGDB_C025492
% Degradation-=92.6%--IKZF2-JurkatEP4660193A1PGDB_A009482PGDB_C025492PGDB_AS002037View
2D structure for PGDB_C025443
% Degradation-=2.4%--IKZF2-JurkatEP4660193A1PGDB_A009801PGDB_C025443PGDB_AS002037View
2D structure for PGDB_C025432
% Degradation-=11%----JurkatEP4660193A1PGDB_A010334PGDB_C025432PGDB_AS000451View
2D structure for PGDB_C025455
Dmax-=100.0%----JurkatEP4660193A1PGDB_A010498PGDB_C025455PGDB_AS000303View
2D structure for PGDB_C025482
% Degradation-=12.2%--IKZF2-JurkatEP4660193A1PGDB_A010519PGDB_C025482PGDB_AS002037View
2D structure for PGDB_C025472
% Degradation-=68.7%--IKZF2-JurkatEP4660193A1PGDB_A010554PGDB_C025472PGDB_AS002037View
2D structure for PGDB_C025465
% Degradation-=91.33%--IKZF2-JurkatEP4660193A1PGDB_A010635PGDB_C025465PGDB_AS002037View
2D structure for PGDB_C025421
% Degradation-=51.9%----JurkatEP4660193A1PGDB_A011601PGDB_C025421PGDB_AS000451View