Summary
AssigneeNovartis
Filing years2019-2025
Patents6
Compounds363
Activity records911
Patent families6
Targets9
Assay familiesbinding, degradation
Activity metricsAC50, DC50, EC50, IC50, degradation
Overview

Target distribution and active-compound trend

Target distribution

911 activity records

9 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0119237202120232025
Activity compounds and values

Activity records

911 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C006511
AC50-=13.1uM-IKZF2-293GTCN113490528APGDB_A007495PGDB_C006511PGDB_AS000852View
2D structure for PGDB_C006501
AC50-=0.079uM-IKZF2-293GTCN113490528APGDB_A007621PGDB_C006501PGDB_AS000852View
2D structure for PGDB_C006513
AC50-=10uM-IKZF2-293GTCN113490528APGDB_A008214PGDB_C006513PGDB_AS000852View
2D structure for PGDB_C006513
% Degradation-=40%--IKZF2-293GTCN113490528APGDB_A009670PGDB_C006513PGDB_AS001176View
2D structure for PGDB_C006496
% Degradation-=80%--IKZF2-293GTCN113490528APGDB_A010504PGDB_C006496PGDB_AS001176View
2D structure for PGDB_C006508
AC50->30uM-IKZF1-293GTCN113490528APGDB_A011148PGDB_C006508PGDB_AS000530View
2D structure for PGDB_C006500
AC50->30uM-IKZF1-293GTCN113490528APGDB_A011484PGDB_C006500PGDB_AS000530View
2D structure for PGDB_C006506
% Degradation-=50%--IKZF2-293GTCN113490528APGDB_A014911PGDB_C006506PGDB_AS001176View
2D structure for PGDB_C006513
AC50->30uM-IKZF1-293GTCN113490528APGDB_A017485PGDB_C006513PGDB_AS000530View
2D structure for PGDB_C006503
% Degradation-=70%--IKZF2-293GTCN113490528APGDB_A017736PGDB_C006503PGDB_AS001176View
2D structure for PGDB_C006507
% Degradation-=74%--IKZF2-293GTCN113490528APGDB_A019674PGDB_C006507PGDB_AS001176View
2D structure for PGDB_C006512
AC50->30uM-IKZF1-293GTCN113490528APGDB_A019954PGDB_C006512PGDB_AS000530View
2D structure for PGDB_C006508
% Degradation-=70%--IKZF2-293GTCN113490528APGDB_A020739PGDB_C006508PGDB_AS001176View
2D structure for PGDB_C006510
% Degradation-=30%--IKZF2-293GTCN113490528APGDB_A021112PGDB_C006510PGDB_AS001176View
2D structure for PGDB_C006514
% Degradation-=40%--IKZF2-293GTCN113490528APGDB_A024698PGDB_C006514PGDB_AS001176View
2D structure for PGDB_C006508
AC50-=2.2uM-IKZF2-293GTCN113490528APGDB_A025125PGDB_C006508PGDB_AS000852View
2D structure for PGDB_C006501
% Degradation-=70%--IKZF2-293GTCN113490528APGDB_A025468PGDB_C006501PGDB_AS001176View
2D structure for PGDB_C006515
AC50-=0.017uM-IKZF2-293GTCN113490528APGDB_A027108PGDB_C006515PGDB_AS000852View
2D structure for PGDB_C006505
AC50->30uM-IKZF1-293GTCN113490528APGDB_A027380PGDB_C006505PGDB_AS000530View
2D structure for PGDB_C006503
AC50-=0.014uM-IKZF2-293GTCN113490528APGDB_A027624PGDB_C006503PGDB_AS000852View