Summary
AssigneeUniversity Of California Berkeley
Filing years2023-2025
Patents2
Compounds108
Activity records122
Patent families2
Targets5
Assay familiesbinding, degradation
Activity metricsDC50, IC50
Overview

Target distribution and active-compound trend

Target distribution

122 activity records

5 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0521032025
Activity compounds and values

Activity records

122 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C007784
DC50->10uM-CDK4--EP4605088A1PGDB_A008016PGDB_C007784PGDB_AS000031View
2D structure for PGDB_C007803
IC50-<100nM-RNF126--EP4605088A1PGDB_A008173PGDB_C007803PGDB_AS000743View
2D structure for PGDB_C007799
IC50-<100nM-RNF126--EP4605088A1PGDB_A008192PGDB_C007799PGDB_AS000743View
2D structure for PGDB_C007772
DC50->10uM-CDK4--EP4605088A1PGDB_A008935PGDB_C007772PGDB_AS000031View
2D structure for PGDB_C007725
DC50->1uM-BRD4--EP4605088A1PGDB_A010072PGDB_C007725PGDB_AS000558View
2D structure for PGDB_C007788
DC50->5uM-SMARCA2--EP4605088A1PGDB_A010493PGDB_C007788PGDB_AS002033View
2D structure for PGDB_C007722
DC50->1uM-BRD4--EP4605088A1PGDB_A011079PGDB_C007722PGDB_AS000558View
2D structure for PGDB_C007771
DC50->10uM-CDK4--EP4605088A1PGDB_A011555PGDB_C007771PGDB_AS000031View
2D structure for PGDB_C007747
DC50->5uM-BRD4--EP4605088A1PGDB_A012397PGDB_C007747PGDB_AS000558View
2D structure for PGDB_C007783
DC50-=1-10uM-CDK4--EP4605088A1PGDB_A012406PGDB_C007783PGDB_AS000031View
2D structure for PGDB_C007798
IC50-<100nM-RNF126--EP4605088A1PGDB_A012516PGDB_C007798PGDB_AS000743View
2D structure for PGDB_C007818
IC50-<100nM-RNF126--EP4605088A1PGDB_A013223PGDB_C007818PGDB_AS000743View
2D structure for PGDB_C007780
DC50-=1-10uM-CDK4--EP4605088A1PGDB_A013311PGDB_C007780PGDB_AS000031View
2D structure for PGDB_C007734
DC50-=0.1-1uM-BRD4--EP4605088A1PGDB_A016101PGDB_C007734PGDB_AS000558View
2D structure for PGDB_C007745
DC50->5uM-BRD4--EP4605088A1PGDB_A016167PGDB_C007745PGDB_AS000558View
2D structure for PGDB_C007795
IC50-=0.1-1uM-RNF126--EP4605088A1PGDB_A016520PGDB_C007795PGDB_AS000743View
2D structure for PGDB_C007777
DC50->10uM-CDK4--EP4605088A1PGDB_A017337PGDB_C007777PGDB_AS000031View
2D structure for PGDB_C007759
DC50->10uM-CDK4--EP4605088A1PGDB_A017408PGDB_C007759PGDB_AS000031View
2D structure for PGDB_C007797
IC50-=0.1-1uM-RNF126--EP4605088A1PGDB_A019177PGDB_C007797PGDB_AS000743View
2D structure for PGDB_C007801
IC50-<100nM-RNF126--EP4605088A1PGDB_A020661PGDB_C007801PGDB_AS000743View