Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C010134
3 activity records1 related patents
2D structure
COC12CC(c3nnc(N[C@H]4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)[C@@H]4C)o3)(C1)C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.4 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025090727A1 | PGDB_A010610 | PGDB_C010134 | PGDB_AS001842 | View |
| Dmax | - | = | 47.5 | % | - | 24 h | CDK2 | - | HEK293 | WO2025090727A1 | PGDB_A037103 | PGDB_C010134 | PGDB_AS002016 | View |
| DC50 | - | = | 785.1 | nM | - | — | CDK2 | - | HEK293 | WO2025090727A1 | PGDB_A051372 | PGDB_C010134 | PGDB_AS001688 | View |