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Compound
PGDB_C012494
4 activity records1 related patents
2D structure
Cn1c(-c2ccc(C3CCOCC3)cc2)cnc1CN1CC[C@H](Oc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ymin | - | = | 36.5 | % | Concentration series: 1 uM, 10 uM | 4 h | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A027372 | PGDB_C012494 | PGDB_AS000656 | View |
| Ymin | - | = | 9.13 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A047964 | PGDB_C012494 | PGDB_AS000093 | View |
| EC50 | - | = | 0.0044 | uM | - | — | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A052864 | PGDB_C012494 | PGDB_AS000951 | View |
| EC50 | - | = | 0.0032 | uM | - | — | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A054203 | PGDB_C012494 | PGDB_AS002574 | View |