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Compound
PGDB_C012535
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(O[C@H]4CCN(Cc5cnn(-c6ccnc(C(F)(F)F)c6)c5)C4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ymin | - | = | 26.36 | % | Concentration series: 1 uM, 10 uM | 4 h | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A023180 | PGDB_C012535 | PGDB_AS000656 | View |
| Ymin | - | = | 16.03 | % | Concentration series: 1 uM, 10 uM | 120 h | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A042361 | PGDB_C012535 | PGDB_AS000093 | View |
| EC50 | - | = | 0.0603 | uM | - | — | WEE1 | - | MKN45 | WO2026030657A1 | PGDB_A058519 | PGDB_C012535 | PGDB_AS002574 | View |
| EC50 | - | = | 0.0126 | uM | - | — | WEE1 | - | LentiX-oeWEE1-ePL | WO2026030657A1 | PGDB_A069465 | PGDB_C012535 | PGDB_AS000951 | View |