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O=C1CCC(N2Cc3cc(CN4CCN(C5CCN(c6ccc(Nc7nnc8nc(Nc9ccccc9)n(C9CCCC9)c8n7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | EGFR | - | THP-1 | CN116239566A | PGDB_A037875 | PGDB_C019598 | PGDB_AS002327 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A062260 | PGDB_C019598 | PGDB_AS000044 | View | |
| IC50 | - | < | 50 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A062522 | PGDB_C019598 | PGDB_AS000044 | View |