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COc1cc(NCc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1000-5000 | nM | - | — | EGFR | - | PC-9 | CN116239566A | PGDB_A031717 | PGDB_C019599 | PGDB_AS000044 | View | |
| IC50 | - | = | 100-500 | nM | - | — | EGFR | - | NCI-H358 | CN116239566A | PGDB_A064146 | PGDB_C019599 | PGDB_AS000770 | View |